Search results for " Clearance"

showing 10 items of 86 documents

Synthesis and evaluation of (S)-2-(2-[18F]fluoroethoxy)-4-([3-methyl-1-(2-piperidin-1-yl-phenyl)-butyl-carbamoyl]-methyl)-benzoic acid ([18F]repaglin…

2004

18F-labeled non-sulfonylurea hypoglycemic agent (S)-2-(2-[(18)F]fluoroethoxy)-4-((3-methyl-1-(2-piperidin-1-yl-phenyl)-butylcarbamoyl)-methyl)-benzoic acid ([(18)F]repaglinide), a derivative of the sulfonylurea-receptor (SUR) ligand repaglinide, was synthesized as a potential tracer for the non-invasive investigation of the sulfonylurea 1 receptor status of pancreatic beta-cells by positron emission tomography (PET) in the context of type 1 and type 2 diabetes. [(18)F]Repaglinide could be obtained in an overall radiochemical yield (RCY) of 20% after 135 min with a radiochemical purity higher than 98% applying the secondary labeling precursor 2-[(18)F]fluoroethyltosylate. Specific activity w…

Fluorine RadioisotopesCancer ResearchBiodistributionMetabolic Clearance RateReceptors DrugContext (language use)Sulfonylurea ReceptorsRats Sprague-DawleyIslets of Langerhanschemistry.chemical_compoundPiperidinesmedicineRadioligandAnimalsTissue DistributionRadiology Nuclear Medicine and imagingPotassium Channels Inwardly RectifyingBenzoic acidChemistryBiological activityLigand (biochemistry)RepaglinideRatsDissociation constantBiochemistryOrgan SpecificityRats Inbred LewIsotope LabelingPositron-Emission TomographyFeasibility StudiesMolecular MedicineATP-Binding Cassette TransportersCarbamatesMultidrug Resistance-Associated ProteinsRadiopharmaceuticalsNuclear chemistrymedicine.drugNuclear Medicine and Biology
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Oxidative stress in ciliated nasal epithelial cells from patients with primary ciliary dyskinesia

2016

Background: Primary ciliary dyskinesia (PCD) is a rare disorder characterized by dysfunction of respiratory cilia and impaired mucociliary clearance leading to recurrent airway infection and chronic inflammation appearing in childhood. Rationale and aims: Chronic inflammation has been associated to oxidative stress (OS). Moreover, evidence of increased OS in the airways of stable children with PCD has been shown (Zihlif, N. et al . Pediatr Pulmonol 2006; 41:509-14). We hypothesize that OS would be increased in ciliated nasal epithelial cells (CNEC) from patients with PCD. This study was aimed to assess the OS profile in CNEC isolated from children with PCD. Methods: CNEC were obtained from …

medicine.medical_specialtyPathologyanimal structuresMucociliary clearancebusiness.industryInflammationGlutathionemedicine.diseasemedicine.disease_causePathophysiologyrespiratory tract diseasesNitric oxidechemistry.chemical_compoundEndocrinologychemistryInternal medicineotorhinolaryngologic diseasesmedicineRespiratory systemmedicine.symptombusinessOxidative stressPrimary ciliary dyskinesia7.1 Paediatric Respiratory Physiology and Sleep
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Endonasal Sinus Surgery Improves Mucociliary Transport in Severe Chronic Sinusitis

1997

A total of 22 patients with extensive chronic sinusitis were examined before and 7.2 ± 1.1 months after microscopic endonasal sinus surgery. Pre- and postoperative nasal mucociliary transport was measured using a modified saccharine test and ciliary beat frequency of nasal respiratory cells using video interference contrast microscopy. In patients suffering from chronic sinusitis, nasal ciliary beat frequency was significantly lower (8.0 ± 1.8 Hz) than in normals (9.5 ± 1.7 Hz, p < 0.02). Following endonasal sinus surgery, ciliary beat frequency in patients with chronic sinusitis remained reduced (8.3 ± 1.2 Hz). Nasal mucociliary transport time was significantly (p < 0.05) longer (20…

AdultMaleTransport timeEpithelium03 medical and health sciences0302 clinical medicineNasal mucusotorhinolaryngologic diseasesRecurrent diseasemedicineHumansMicroscopy InterferenceIn patientCiliaSinusitisRespiratory system030223 otorhinolaryngologyMicroscopy Videomedicine.diagnostic_testbusiness.industryChronic sinusitisEndoscopyMiddle AgedSinus surgeryEndoscopyOtorhinolaryngologyMucociliary Clearance030220 oncology & carcinogenesisAnesthesiaChronic DiseaseFemalebusinessAmerican Journal of Rhinology
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Effect of salinity and temperature on feeding physiology and scope for growth of an invasive species (Brachidontes pharaonis - MOLLUSCA: BIVALVIA) wi…

2008

Abstract The Indo-Pacific mytilid Brachidontes pharaonis (Bivalvia, Fischer 1870) offers an excellent model for the study of “Lessepsian migration” and the successive colonization at new Mediterranean locations. This species in out competing indigenous bivalves is particularly well adapted to Mediterranean conditions and this is likely due to biological characteristics and physio-ecological plasticity. In the present paper, we report on clearance rate (CR), respiration rate (RR) and Scope for Growth (SFG) of B. pharaonis collected from a Western Sicilian pond (Southern Tyrrhenian, MED). Physiological variables were determined in response to a range of temperatures from 11 ° to 20 °C and a b…

Settore BIO/07 - EcologiaLessepsian migrationEcologyAquatic ScienceBiologybiology.organism_classificationBivalviaBiological invasions Brachidontes pharaonis Clearance rate Lesseptian migration Mediterranean Scope for growthSalinityMediterranean seaBrachidontes pharaonisRespiration rateClearance rateMolluscaEcology Evolution Behavior and SystematicsJournal of Experimental Marine Biology and Ecology
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Performance Comparison of Alternative Hollow-Fiber Modules for Hemodialysis by Means of a CFD-Based Model

2022

Commercial hemodialyzers are hollow-fiber cylindrical modules with dimensions and inlet–outlet configurations dictated mostly by practice. However, alternative configurations are possible, and one may ask how they would behave in terms of performance. In principle, it would be possible to depart from the standard counter-flow design, while still keeping high clearance values, thanks to the increase in the shell-side Sherwood number (Sh) due to the cross-flow. To elucidate these aspects, a previously developed computational model was used in which blood and dialysate are treated as flowing through two interpenetrating porous media. Measured Darcy permeabilities and mass transfer coefficients…

Settore ING-IND/26 - Teoria Dello Sviluppo Dei Processi ChimiciSettore ING-IND/25 - Impianti ChimiciProcess Chemistry and TechnologyPorous mediaHollow-fiber membraneUltrafiltrationhemodialysis; hollow-fiber membrane; solute clearance; computational fluid dynamics; porous media; Darcy permeability; ultrafiltration; mass transferFiltration and SeparationComputational fluid dynamicsHemodialysisChemical Engineering (miscellaneous)Mass transferDarcy permeabilitySettore ING-IND/19 - Impianti NucleariSolute clearanceMembranes
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Effect of acyl-CoA oxidase activity on the accumulation of gamma-decalactone by the yeast Yarrowia lipolytica: a factorial approach.

2007

International audience; beta-Oxidation is a cyclic pathway involved in the degradation of lipids. In yeast, it occurs in peroxisomes and the first step is catalyzed by an acyl-CoA oxidase (Aoxp). The yeast Yarrowia lipolytica possesses several genes (POX) coding for Aoxps. This study is based on the factorial analysis of results obtained with the many POX derivative strains that have been constructed previously. The effect of interactions between Aoxps on the acyl-CoA oxidase (Aox) activity was important even at the second order. We then investigated the effect of Aox activity on growth and lactone production. Aox activity was correlated with acidification of the medium by cells and with ce…

0106 biological sciencesYarrowia lipolyticaMESH: Enzyme ActivationMetabolic Clearance RateMESH: Factor Analysis StatisticalYarrowiaBiologymodèleModels Biological01 natural sciencesApplied Microbiology and BiotechnologyLactones03 medical and health sciencesEnzyme activatorSpecies SpecificityMESH: Computer Simulation010608 biotechnologyCombinatorial Chemistry TechniquesAcyl-CoA oxidaseMESH: Species SpecificityComputer Simulation030304 developmental biologychemistry.chemical_classificationMESH: Metabolic Clearance Rate0303 health sciencesOxidase testmétabolisme des acides grasAcyl-CoA oxidase activityMESH: Acyl-CoA OxidaseMESH: Models BiologicalYarrowia[SDV.BBM.BM]Life Sciences [q-bio]/Biochemistry Molecular Biology/Molecular biologyGeneral MedicinePeroxisomebiology.organism_classificationYeastEnzyme ActivationBiochemistrychemistrylactoneMolecular MedicineMESH: Combinatorial Chemistry TechniquesMESH: YarrowiaAcyl-CoA OxidaseFactor Analysis StatisticalLactoneMESH: Lactones
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Gadolinium accumulation after contrast-enhanced magnetic resonance imaging: Which implications in patients with Crohn's disease?

2017

Crohn's disease (CD) is a chronic inflammatory condition of the bowel, characterized by an alternation of remission and relapse phases, leading to a progressive intestinal damage with loss of function. Magnetic resonance enterography has been widely used in the past for the evaluation of fistulizing disease, but its use increased over time, being considered helpful in different moments of disease course. Intravenous injection of Gadolinium-based contrast agents has been demonstrated to be crucial to assess mucosal inflammation, transmural involvement, and extraintestinal disease. Recently, Gadolinium accumulation in human tissues has been increasingly reported, although clinical implication…

medicine.medical_specialtyPathologyMetabolic Clearance RateGadoliniumchemistry.chemical_elementContrast MediaGadoliniumDiseaseGastroenterology030218 nuclear medicine & medical imaging03 medical and health sciencesGadolinium storage condition0302 clinical medicineCrohn DiseaseInternal medicineMedicineHumansIn patientTissue DistributionContrast-enhanced Magnetic Resonance ImagingCrohn's diseasemedicine.diagnostic_testHepatologybusiness.industryCrohn's disease; Gadolinium; Gadolinium storage condition; Magnetic resonance imaging; Hepatology; GastroenterologyGastroenterologyMagnetic resonance imagingHepatologymedicine.diseaseMagnetic resonance enterographyMagnetic Resonance ImagingCrohn's diseasechemistryDisease Progression030211 gastroenterology & hepatologybusinessDigestive and liver disease : official journal of the Italian Society of Gastroenterology and the Italian Association for the Study of the Liver
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Human hepatic cell uptake of resveratrol: involvement of both passive diffusion and carrier-mediated process

2004

This work reports significant advances on the transport in hepatic cells of resveratrol, a natural polyphenol with potent protective properties. First, we describe a new simple technique to qualitatively follow resveratrol cell uptake and intracellular distribution, based on resveratrol fluorescent properties. Second, the time-course study and the quantification of (3)H-labelled resveratrol uptake have been performed using human hepatic derived cells (HepG2 tumor cells) and hepatocytes. The temperature-dependence of the kinetics of uptake as well as the cis-inhibition experiments agree with the involvement of a carrier-mediated transport in addition to passive diffusion. The decrease of pas…

HepatoblastomaMetabolic Clearance RateCellBiophysicsBiological AvailabilityBiological Transport ActiveResveratrolBiochemistryCell LineDiffusionchemistry.chemical_compoundResveratrol bindingCell Line TumorStilbenesmedicineHumansDistribution (pharmacology)Tissue DistributionMolecular BiologyTemperaturefood and beveragesCell BiologyBlood proteinsmedicine.anatomical_structurechemistryBiochemistryResveratrolCell cultureHepatocytesHepatic stellate cellBiophysicsCarrier ProteinsIntracellularBiochemical and Biophysical Research Communications
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Regional blood flow in deep structures of the brain measured in acute cat experiments by means of a new beta-sensitive semiconductor needle detector.

1967

Regional cerebral blood flow was measured by means of isotope clearance with a new type of solid state beta-sensitive needle detector (diameter 0.9 mm) introduced into the brain tissue in acute cat experiments. The flow values obtained within the cortex were compared with values recorded above the same cortical region with the same needle detector, or with a small GM-tube. The insertion of the needle detector into the brain tissue gave rise to injury (checked histologically) which deformed the clearance curves in a manner suggesting that the normal circulation had been destroyed within the tissue from which the measurements were made.

Materials scienceMetabolic Clearance RateSolid-stateBlood PressureBrain EdemaCortex (anatomy)medicineAnimalsBeta (finance)Cerebral CortexRadioisotopesIsotopebusiness.industryGeneral NeuroscienceDetectorKryptonBlood flowSemiconductormedicine.anatomical_structureCerebral blood flowSemiconductorsRegional Blood FlowCerebrovascular CirculationCatsbusinessNuclear medicineBlood Flow VelocityBiomedical engineeringExperimental brain research
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Prevalence and severity of anaemia in patients with type 2 diabetic nephropathy and different degrees of chronic renal insufficiency.

2007

<i>Background/Aim:</i> Type 2 diabetes mellitus is the single most common cause of chronic kidney disease (CKD); however its real impact on renal anaemia has not been established. The aim of this study was to evaluate whether onset, severity, and prevalence of anaemia during the course of CKD is different between type 2 diabetic and non-diabetic patients. <i>Methods:</i> We enrolled 281 patients with: (1) type 2 diabetes and no CKD (n = 75); (2) type 2 diabetes plus CKD (n = 106), and (3) CKD without type 2 diabetes (n = 100). According to K/DOQI guidelines, the patients with renal insufficiency (i.e., those with a glomerular filtration rate <60 ml/min) were subgr…

NephrologyMaleglomerulus filtration rateType 2 diabetesurologic and male genital diseasesGastroenterologySeverity of Illness Indexadult; aged; anemia; article; chronic kidney failure; comparative study; controlled study; creatinine clearance; diabetic nephropathy; disease course; disease severity; female; glomerulus filtration rate; hemoglobin blood level; human; kidney failure; kidney function; major clinical study; male; non insulin dependent diabetes mellitus; practice guideline; prevalence; priority journal; risk assessment; Aged; Anemia; Creatinine; Diabetes Mellitus Type 2; Diabetic Nephropathies; Female; Glomerular Filtration Rate; Hemoglobins; Humans; Kidney Failure Chronic; Male; Middle Aged; Prevalence; Severity of Illness Index; Sex DistributionKidney FailureDiabetic nephropathychemistry.chemical_compoundHemoglobinsChronic kidney diseasecreatinine clearancePrevalenceDiabetic NephropathiesChronickidney functioncomparative studynon insulin dependent diabetes mellitusadultdisease coursearticlerisk assessmentAnemiaGeneral Medicinechronic kidney failureMiddle Agedpriority journalNephrologyCreatininedisease severityFemaleType 2Glomerular Filtration Ratemedicine.medical_specialtyAnaemia diabetes mellitus; Chronic kidney disease diabetes mellitus; Type 2 diabetes mellitus anaemiaRenal functionAnaemiaDiabetes mellitusInternal medicineType 2 diabetes mellitusDiabetes MellitusmedicineHumanscontrolled studyhumanSex DistributionAgedSettore MED/14 - NefrologiaCreatininehemoglobin blood levelbusiness.industrydiabetic nephropathypractice guidelineType 2 Diabetes Mellitusmedicine.diseasemajor clinical studySurgerychemistryDiabetes Mellitus Type 2Kidney Failure ChronicbusinessKidney disease
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